체외 평가
체외시험에 의해 합성된 화합물에 의한 젤라틴 효소의 억제활성효소 분석과 젤라틴 효소 스펙트럼과 같은 기술은 그들의 유효성을 측정하는 데 사용될 수 있다.젤라틴 효소가 억제하는 아나몰 범위 내에 있어야 하는 IC50 값을 결정해야 합니다.
화학 원료를 구입해야하는 경우 요청 정보를 제출하여최신견적을받으십시오.
체외 평가의 학술 논문
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Design, Synthesis, and Biological Evaluation of Tetrahydro-β-carboline Derivatives as Selective Sub-Nanomolar Gelatinase Inhibitors
화학 물질
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(1RS)-2-(4''-methoxy-4'-phenoxybenzenesulfonyl)-1,2,3,4-tetrahydro-norarmano-1-carboxylic acid
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Synthesis and evaluation of β-carboline derivatives as potential monoamine oxidase inhibitors
화학 물질
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7-(phenethoxy)-1-methyl-β-carboline
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Design, synthesis, and biological evaluation of new raloxifene analogues of improved antagonist activity and endometrial safety
화학 물질
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(4-(2-hydroxyethoxy)phenyl)(6-methoxy-2-(4-methoxyphenyl)benzo[b]thiophen-3-yl)methanone
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Synthesis, in vitro, and in vivo evaluation of phosphate ester derivatives of combretastatin A-4
화학 물질
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diisopropyl-phosphoramidous acid 2-cyano-ethyl ester cyclohexyl ester
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New fluorinated dopamine D2 ligands with benzofuran skeleton. The synthesis and in vitro evaluation
화학 물질
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7-carboxy-5-ethyl-2,3-dihydrobenzofuran
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Synthesis, in vitro and in vivo evaluation of novel substituted N-(4-(2-(4-benzylpiperazin-1-yl)ethoxy)phenyl)-N-methyl-quinazolin-4-amines as potent antitumor agents
화학 물질
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1-(2-Chloroethyl)-4-[(2-fluorophenyl)methyl]piperazine
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Synthesis and in vitro evaluation of xylene linked carbamoyl bis-pyridinium monooximes as reactivators of organophosphorus (OP) inhibited electric eel acetylcholinesterase (AChE)
화학 물질
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1-(2-bromomethylbenzyl)-3-hydroxyiminomethylpyridinium bromide
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Design, synthesis, and in vitro evaluation of aza-peptide aldehydes and ketones as novel and selective protease inhibitors
화학 물질
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L-Alanine, N-[(phenylmethoxy)carbonyl]-L-alanyl-, hydrazide
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Towards to hENT1-nucleoside transporter selective imaging agents. Synthesis and in vitro evaluation of the radiolabeled SAENTA analogues
화학 물질
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12,13-Dithia-2,9,16,23-tetraazatetracosanedioic acid, 8,17-dioxo-, bis(1,1-dimethylethyl) ester
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Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) Family
화학 물질
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Propanedioic acid, methyl-, monoethyl ester, potassium salt
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Synthesis and in vitro evaluation of tetrahydroisoquinolinyl benzamides as ligands for σ receptors
화학 물질
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4-(3,4-dimethoxyphenethylamino)butanenitrile
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