약리 활성
타듐술폰아미드계 화합물은 5-HT2 수용체의 길항제로 연구된 바 있다.이 수용체들은 감정, 인지, 중추신경계를 조절하는 다른 과정에 관여한다.길항제는 이들 수용체와 결합하고 5-히드록시셀아민을 통해 이들의 활성화를 억제하는데, 5-하이드록시셀라민은 표적의 5-HT2 수용체의 특정 아형에 따라 다른 효과를 낼 수 있다.
화학 원료를 구입해야하는 경우 요청 정보를 제출하여최신견적을받으십시오.
약리 활성의 학술 논문
-
Naphthosultam Derivatives: A New Class of Potent and Selective 5-HT2 Antagonists
화학 물질
-
2-<3-(4-phenyl-1,2,3,6-tetrahydropyridyl)propyl>-2H-naphth<1,8-cd>isothiazole 1,1-dioxide
-
-
SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF GUANIDINE AND 2-AMINO 2-IMIDAZOLINE DERIVATIVES
화학 물질
-
1-(2,6-Dichlorophenyl)-2-dimethylaminoimidazolines
-
-
Synthesis and structure-activity relationship of spiro[isochromanpiperidine]analogues for inhibition of histamine release
화학 물질
-
1'-phenethyl-spiro[isochroman-4,4'-piperidine]; hydrochloride
-
-
SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF 4-ARYL-1,4-DIHYDROPYRIDINES
화학 물질
-
diethyl 2,6-dimethyl-4-[2-(trifluoromethyl)phenyl]-1,4-dihydropyridine-3,5-dicarboxylate
-
-
Synthesis and Characterization of Selected Heteroarotinoids. Pharmacological Activity as Assessed in Vitamin A Deficient Hamster Tracheal Organ Cultures. Single-Crystal X-ray Diffraction Analysis of 4,4-Dimethylthiochroman-6-yl Methyl Ketone 1,1-Dioxide and Ethyl (E)-p-<2-(4,4-Dimeth...
화학 물질
-
4-[(Z)-2-(4,4-Dimethyl-chroman-6-yl)-propenyl]-benzoic acid ethyl ester
-
-
Anti-inflammatory activity of substituted 1,3,4-oxadiazoles
화학 물질
-
2-[(biphenyl-4-yloxy)acetyl]-N-phenylhydrazinecarbothioamide
-
-
4-Amino-6-chloro-2-piperazinopyrimidines with selective affinity for α2-adrenoceptors
화학 물질
-
6-chloro-5-methyl-2-(piperazin-1-yl)-N-(propan-2-yl)pyrimidin-4-amine
-
-
Central pharmacological activity of a new piperazine derivative: 4-(1-Phenyl-1h-pyrazol-4-ylmethyl)-piperazine-1-carboxylic acid ethyl ester
화학 물질
-
4-(1-phenyl-(1H-pyrazol-4-ylmethyl))-piperazine-1-carboxylic acid ethyl ester
-
