억제
생물학적 활성이나 효소 반응을 막거나 차단하는 과정입니다.
화학 원료를 구입해야하는 경우 요청 정보를 제출하여최신견적을받으십시오.
억제의 학술 논문
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Synthesis and evaluation of tricyclic pyrrolopyrimidinones as dipeptide mimetics: Inhibition of interleukin-1β-converting enzyme
화학 물질
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(S)-1-(2-Azido-benzoyl)-5-oxo-pyrrolidine-2-carboxylic acid tert-butyl ester
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Synthesis and Inhibition of Human Acrosin and Trypsin and Acute Toxicity of Aryl 4-Guanidinobenzoates
화학 물질
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4-Guanidino-benzoic acid 3-cyano-phenyl ester; hydrochloride
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Discovery of multifunctional anti-Alzheimer's agents with a unique mechanism of action including inhibition of the enzyme butyrylcholinesterase and γ-aminobutyric acid transporters
화학 물질
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(2R,3S)-3-amino-1-((3-(tert-butyl)benzyl)amino)-4-phenylbutan-2-ol
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Nucleomimetic strategy for the inhibition of HIV-1 nucleocapsid protein NCp7 activities
화학 물질
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thiocarbonic acid O-[2-(tert-butyl-diphenyl-silanyloxymethyl)-5-(5-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-tetrahydro-furan-3-yl] ester O-p-tolyl ester
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Inhibition of human neutrophil elastase with peptidyl electrophilic ketones. 2. Orally active p(G)-Val-Pro-Val pentafluoroethyl ketones
화학 물질
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1(RS)-N-[4-[N-(4-Chlorophenylsulfonyl)carbamoyl]benzoyl]-L-valyl-N-[2-methyl-1-(trifluoroacetyl)propyl]-L-prolinamide
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Inhibition of DNA topoisomerase II by azaelliptitoxins functionalized in the variable substituent domain
화학 물질
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Carbonic acid benzyl ester 2,6-dimethoxy-4-((3aR,4R,10R)-4-methoxy-1-oxo-3a,4,9,10-tetrahydro-3H-2-oxa-9,10a-diaza-cyclopenta[b]fluoren-10-yl)-phenyl ester
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Nucleomimetic strategy for the inhibition of HIV-1 nucleocapsid protein NCp7 activities
화학 물질
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thiocarbonic acid O-[2-(tert-butyl-diphenyl-silanyloxymethyl)-5-(5-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-tetrahydro-furan-3-yl] ester O-p-tolyl ester
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Inhibition of cyclic adenosine-3',5'-monophosphate phosphodiesterase from vascular smooth muscle by rolipram analogues
화학 물질
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Butanoic acid,4-[2-methoxy-5-(5-oxo-3-pyrrolidinyl)phenoxy]-
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Synthesis and structure-activity relationship of spiro[isochromanpiperidine]analogues for inhibition of histamine release
화학 물질
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1'-phenethyl-spiro[isochroman-4,4'-piperidine]; hydrochloride
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TPA-induced up-regulation of activator protein-1 can be inhibited or enhanced by analogs of the natural product curcumin
화학 물질
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2-Propen-1-one, 1-(2,4-dimethylphenyl)-3-phenyl-
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Inhibition of human enterovirus 71 replication by pentacyclic triterpenes and their novel synthetic derivatives
화학 물질
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methyl 2-O-phenyglycylurs-3,23-isopropylidenedioxyurs-12-ene-28-oate
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An Acyl-Iminium Ion Cyclization Route to a Novel Conformationally Restricted Dipeptide Mimic: Applications to Angiotensin-Converting Enzyme Inhibition
화학 물질
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(4S,7S,12bR)-7-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-6-oxo-1,2,3,4,6,7,8,12b-octahydro-benzo[c]pyrido[1,2-a]azepine-4-carboxylic acid benzhydryl ester
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Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties
화학 물질
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4-nitro-N-(3-phenylpropyl)benzamide
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Synthesis and antiviral activity of 9-alkoxypurines. 1. 9-(3-Hydroxypropoxy)- and 9-[3-hydroxy-2-(hydroxymethyl)propoxy]purines
화학 물질
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2-amino-9-[3-hydroxy-2-(hydroxymethyl)propoxy]-3,9-dihydro-6H-purin-6-one
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Inhibition of ribosomal peptidyltransferase with 2'(3')-O-acetyl-2 inches(3 inches)-O-glycyl-1,2-di(adenosin-N6-yl)ethane and -1,4-di(adenosin-N6-yl)butane. Effect of alkyl chain length.
화학 물질
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9-<2',3'-O-<<
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Inhibition of the tissue factor/factor VIIa complex - Lead optimisation using combinatorial chemistry
화학 물질
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Acetic acid, [4-[[[(4-nitrophenoxy)carbonyl]oxy]methyl]phenoxy]-, 2-propenyl ester
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Inhibition of human leukocyte elastase. 1. Inhibition by C-7-substituted cephalosporin tert-butyl esters
화학 물질
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(6R,7S)-3-Acetoxymethyl-7-benzyloxy-5,5,8-trioxo-5λ6-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid tert-butyl ester
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Inhibition of human leukocyte elastase by N-substituted peptides containing α,α-difluorostatone residues at P1
화학 물질
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Glycine, N-(2,3-dihydro-1H-inden-2-yl)-N-[N-[(phenylmethoxy)carbonyl]-L-valyl]-, ethyl ester
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Design, synthesis and discovery of 2(1H)-quinolone derivatives for the treatment of pulmonary fibrosis through inhibition of TGF-β/smad dependent and independent pathway
화학 물질
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4-(4-aminophenoxy)quinolin-2(1H)-one
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Synthesis of Carbapenems Containing Peptidoglycan Mimetics and Inhibition of the Cross-Linking Activity of a Transpeptidase of l,d Specificity
화학 물질
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Hexanoic acid, 6-[[[(4-nitrophenyl)methoxy]carbonyl]amino]-
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Dehydroalanine-based inhibition of a peptide epimerase from spider venom.
화학 물질
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(S)-tert-butyl 2-((S)-2-(((benzyloxy)carbonyl)amino)-3-phenylpropanamido)propanoate
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Synthesis of 5′-methylenearisteromycin and its 2-fluoro derivative with potent antimalarial activity due to inhibition of the parasite S-adenosylhomocysteine hydrolase
화학 물질
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(3S,4R,5S,6R)-3-ethoxycarbonyloxy-7-[(4-methoxyphenyl)diphenylmethoxy]-4,5-(p-methoxybenzylidenedioxy)-6-(imidazolylthiocarbonyloxy)heptyne
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Inhibition of mitosis by glycopeptide dendrimer conjugates of colchicine
화학 물질
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O-(2,3,4,6-tetra-O-benzyl-α-D-galactopyranosyl)-N-oxyphthalimide
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Chemoselective regulation of TREK2 channel: Activation by sulfonate chalcones and inhibition by sulfonamide chalcones
화학 물질
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4'-(4-aminobenzenesulfonamide)-4-hydroxychalcone
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Pd/PTABS: Catalyst for Room Temperature Amination of Heteroarenes
화학 물질
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2-chloro-4-(4-tosylpiperazin-1-yl)pyrimidine
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The squalestatins: Synthesis and biological activity of some C3-modified analogues; replacement of a carboxylic acid or methyl ester with an isoelectronic heterocyclic functionality
화학 물질
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(1S,3R,4S,5R,6R,7R)-1-((4S,5R)-4-Acetoxy-5-methyl-3-methylene-6-phenyl-hexyl)-4,6,7-trihydroxy-3-(5-methyl-4H-[1,2,4]triazol-3-yl)-2,8-dioxa-bicyclo[3.2.1]octane-4,5-dicarboxylic acid dimethyl ester
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Reactions of a platinum(II) agostic complex: Decyclometalation, dicyclometalation, and solvent-switchable formation of a rollover complex
화학 물질
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[(2-tert-butyl-6-(4-fluorophenyl)pyridine(-2H))Pt(PPh3)]
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Synthesis of substituted triazolyl curcumin mimics that inhibit RANKL-induced osteoclastogenesis
화학 물질
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(E)-1-(3-azidophenyl)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-one
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Synthesis of sialyl Lewis X mimetics and related structures using the glycosyl phosphite methodology and evaluation of E-selectin inhibition
화학 물질
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1H-Pyrrole-1,2-dicarboxylic acid, 2,5-dihydro-, 2-ethyl 1-(phenylmethyl) ester, (R)-
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2-aminobenzimidazole derivatives strongly inhibit and disperse Pseudomonas aeruginosa biofilms
화학 물질
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5-IODO-1H-BENZIMIDAZOLE-2-AMINE
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Proton-Transfer Reactions. 4. Near-Unity Kinetic Isotope Effects for Hydron Exchange and Dehydrofluorination Reactions
화학 물질
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[2,2,2-트리플루오로-1-(트리플루오로메틸)에틸]벤젠
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Inhibition of human alcohol dehydrogenases by formamides
화학 물질
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포름아미드, N-시클로펜틸-N-시클로프로필-(9CI)
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Inhibition of gastric H+, K+-ATPase by novel thiazolidinone derivatives
화학 물질
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3-(3-methylbenzyl)-5-((5-(4-chlorophenyl)furan-2-yl)methylene)thiazolidine-2,4-dione
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Synthesis and evaluation of α-glucosidase and pancreatic lipase inhibition by quinazolinone-coumarin hybrids
화학 물질
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2-(4-fluorobenzyl)quinazolin-4(3H)-one
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Intriguing structure-activity relations underlie the potent inhibition of HIV protease by norstatine-based peptides
화학 물질
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N~1~-{(2S,3S)-4-[(2S)-2-(tert-butylcarbamoyl)pyrrolidin-1-yl]-3-hydroxy-4-oxo-1-phenylbutan-2-yl}-N~2~-[(naphthalen-1-yloxy)acetyl]-L-aspartamide
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Inhibition of urease activity by dipeptidyl hydroxamic acids
화학 물질
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Glycinamide, N-[(1,1-dimethylethoxy)carbonyl]-O-(phenylmethyl)-L-seryl-N-hydroxy-
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