대사 안정성
수식은 이들 화합물의 대사 안정성을 강화시켜 더 긴 반감기와 개선된 약대역학으로 이어질 수 있다.
화학 원료를 구입해야하는 경우 요청 정보를 제출하여최신견적을받으십시오.
대사 안정성의 학술 논문
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SYNTHESIS AND BIOLOGICAL ACTIVITY OF 7,8-SUBSTITUTED THEOPHYLLINES
화학 물질
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1,3-Dimethyl-8-piperidin-1-yl-7-{2-[piperidin-(2Z)-ylideneamino]-ethyl}-3,7-dihydro-purine-2,6-dione
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Design and synthesis of an orally active GPIIb/IIIa antagonist based on a phenylpiperazine scaffold
화학 물질
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tert-Butyl 3-{4-[4-(4-amidinophenyl)-1-piperazinyl]phenyl}propionate
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클로로 벤젠
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Novel sulfamoyl benzamides as selective CB2 agonists with improved in vitro metabolic stability
화학 물질
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4-메틸-3-(4-모르폴리노설포닐)아닐린
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CYP2C9 structure-metabolism relationships: Optimizing the metabolic stability of COX-2 inhibitors
화학 물질
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1H-Pyrazole-3-carboxylic acid, 1-[4-(aminosulfonyl)phenyl]-5-(4-methylphenyl)-, ethyl ester
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Achiral oligoamines as versatile tool for the development of aspartic protease inhibitors
화학 물질
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bis[3-(benzenesulfonylamino)propyl]carbamic acid tert-butyl ester
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Identification of 4-amino-2-cyclohexylaminoquinazolines as metabolically stable melanin-concentrating hormone receptor 1 antagonists
화학 물질
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[4-(1,3-dioxo-1,3-dihydro-isoindol-2-ylmethyl)-cyclohexyl]-carbamic acid tert-butyl ester
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Structure-based design, synthesis, and biological evaluation of irreversible human rhinovirus 3C protease inhibitors. 3. Structure-activity studies of ketomethylene-containing peptidomimetics
화학 물질
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(R)-2-Benzyl-3-((S)-2-benzyloxycarbonylamino-3,3-dimethyl-butyryl)-succinic acid 4-tert-butyl ester 1-methyl ester
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Stereocontrolled Synthesis of Tetrafluoropentanols: Multivicinal Fluorinated Alkane Units for Drug Discovery
화학 물질
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(R)-4-((2R,3S)-3-((benzyloxy)methyl)oxiran-2-yl)-2,2-dimethyl-1,3-dioxolane
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Structure-activity relationships of arylbenzofuran H3 receptor antagonists
화학 물질
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4-(3-bromo-2-{2-[(2R)-2-methylpyrrolidin-1-yl]ethyl}-1-benzofuran-5-yl)benzonitrile
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Enhancing the Cell Permeability and Metabolic Stability of Peptidyl Drugs by Reversible Bicyclization
화학 물질
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methyl 3,5-bis[(acetylsulfanyl)methyl]benzoate
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Synthesis, biological evaluation and molecular docking studies of novel quinazolinones as antitubercular and antimicrobial agents
화학 물질
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2-methylsulfanyl-3-(4-chlorophenyl)-3H-quinazolin-4-one
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Synthesis and anticonvulsant activity of new 2,3-benzodiazepines as AMPA receptor antagonists
화학 물질
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7,8-Methylenedioxy-3-methyl-1-phenyl-3,5-dihydro-2,3-benzodiazepin-4(4H)-one
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1-Substituted vinyl-1-phthalanpropylamines as potential antidepressant agents.
화학 물질
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1,3-디히드로-3,3-디메틸-1-페닐이소벤조푸란-1-올
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A novel class of nonpeptidic biaryl inhibitors of human cathepsin K
화학 물질
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1-(4-BROMO-PHENYL)-4-METHYL-PIPERAZINE
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Synthesis and antiviral properties of spirocyclic [1,2,3]-Triazolooxazine nucleosides
화학 물질
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1-(3-bromoprop-1-yn-1-yl)-3-fluorobenzene
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Sulfonyl fluoride inhibitors of fatty acid amide hydrolase
화학 물질
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1-(4-methoxyphenyl)-7-phenoxyheptane
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Synthesis, conformation and antiviral activity of nucleoside analogues with the (2-hydroxy-1-phenylethoxy)methyl glycone - A family of nucleoside analogues related to d4T and aciclovir
화학 물질
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(S)-[2-(methoxymethoxy)-2-phenyl]ethyl benzoate
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Identification of a new biaryl scaffold generating potent renin inhibitors
화학 물질
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1,3-dichloro-2-{2-[4-(iodomethyl)phenoxy]ethoxy}-5-methylbenzene
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Design, synthesis, and biological evaluation of novel diarylalkyl amides as TRPV1 antagonists
화학 물질
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(E)-N-(3-fluoro-4-(methylsulfonamido)benzyl)-3-(4-iodophenyl)acrylamide
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PK/PD Disconnect Observed with a Reversible Endothelial Lipase Inhibitor
화학 물질
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(SS,E)-N-(3-(3,4-dichlorophenyl)propylidene)-2-methylpropane-2-sulfinamide
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GluN2B-selective N-methyl-d-aspartate (NMDA) receptor antagonists derived from 3-benzazepines: Synthesis and pharmacological evaluation of benzo[7]annulen-7-amines
화학 물질
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methyl 3-acetamido-5-(3-methoxyphenyl)pentanoate
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