생물학적 이용도
체내 활성은 화합물이 체내에서 효과적으로 흡수, 분포, 대사 및 배설될 것을 요구한다.화합물의 약대역학 특성에 영향을 줄 수 있는 발색단을 포함하는 화학구조
화학 원료를 구입해야하는 경우 요청 정보를 제출하여최신견적을받으십시오.
생물학적 이용도의 학술 논문
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Potential antitumor agents. 54. Chromophore requirements for in vivo antitumor activity among the general class of linear tricyclic carboxamides
화학 물질
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N-[2-(dimethylamino)ethyl]phenazine-1-carboxamide
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A selective de-O-methylation of guaiacyl lignans to corresponding catechol derivatives by 2-iodoxybenzoic acid (IBX). the role of the catechol moiety on the toxicity of lignans
화학 물질
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(7,9'-epoxylignan-3,3',4,4',9-pentayl)pentaacetate
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Nonpeptide renin inhibitors with good intraduodenal bioavailability and efficacy in dog
화학 물질
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(2S,4S,5S)-5-{(S)-2-[(S)-1-Benzyl-2-(4-methoxymethoxy-piperidin-1-yl)-2-oxo-ethoxy]-hexanoylamino}-6-cyclohexyl-4-hydroxy-2-isopropyl-hexanoic acid {3-[(imidazole-1-carbothioyl)-amino]-propyl}-amide
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Synthesis and hypoglycemic effect of chrysin derivatives
화학 물질
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chrysin dimethylether
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Structure-cytotoxic activity relationship for the toad poison bufadienolides
화학 물질
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bufalin 3-[N-(tert-butoxycarbonyl)hydrazido]succinate
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4-[1-(4-Fluorobenzyl)-4-hydroxy-1H-indol-3-yl]-2-hydroxy-4-oxobut-2-enoic acid as a prototype to develop dual inhibitors of HIV-1 integration process
화학 물질
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4-[1-(3,5-dimethylbenzyl)-4-methoxy-1H-indol-3-yl]-2-hydroxy-4-oxobut-2-enoic acid
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Synthesis and evaluation of inhibitors of cytochrome P450 3A (CYP3A) for pharmacokinetic enhancement of drugs
화학 물질
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bis-N-[(S)-2-(pyrazol-4-ylmethoxycarbonylamino)-3-phenylpropyl]ethylamine
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2-Arylmethylaminomethyl-5,6-dihydroxychromone derivatives with selective anti-HCV activity
화학 물질
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acetic acid 2-acetyl-4-benzyloxy-3-methoxy-phenyl ester
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Synthesis and antiviral properties of spirocyclic [1,2,3]-Triazolooxazine nucleosides
화학 물질
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1-(3-bromoprop-1-yn-1-yl)-3-fluorobenzene
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Ramberg-Backlund rearrangement vs. β-Elimination of haloform from trichloro and trifluoromethyl sulfones
화학 물질
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Diphenylmethyl-dichlormethyl-sulfon
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Hypocholesterolemic Activity of Synthetic and Natural Tocotrienols
화학 물질
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3,4-dihydro-6-<(2-methoxyethoxy)methoxy>-2,5,7,8-tetramethyl-2-<6-<(4-methylphenyl)sulfonyl>-4,8,12-trimethyltrideca-3(E),7(E),11-trienyl>-2H-1-benzopyran
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Design, synthesis, and bioavailability evaluation of coumarin-based prodrug of meptazinol
화학 물질
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Propionic acid 2-((Z)-3-hydroxy-propenyl)-phenyl ester
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Synthesis, biological evaluation and molecular docking studies of novel quinazolinones as antitubercular and antimicrobial agents
화학 물질
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2-methylsulfanyl-3-(4-chlorophenyl)-3H-quinazolin-4-one
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Structure-based discovery of pyrazolobenzothiazine derivatives as inhibitors of hepatitis C virus replication
화학 물질
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methyl 1-(4-fluorophenyl)-4-methyl-1,4-dihydropyrazolo[4,3-c][1,2]benzothiazine-3-carboxylate 5,5-dioxide
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A novel class of nonpeptidic biaryl inhibitors of human cathepsin K
화학 물질
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1-(4-BROMO-PHENYL)-4-METHYL-PIPERAZINE
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Ultra-Short-Acting β-Adrenergic Receptor Blocking Agents. 2. (Aryloxy)propanolamines Containing Esters on the Aryl Function
화학 물질
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2-Propenoic acid, 3-[4-(oxiranylmethoxy)phenyl]-, methyl ester
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Bifunctional acyclic nucleoside phosphonates: 2. Symmetrical 2-{[bis(phosphono)methoxy]methyl}ethyl derivatives of purines and pyrimidines
화학 물질
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5-[(benzyloxy)methyl]-2,2-dimethyl-1,3-dioxane
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Synthesis, conformation and antiviral activity of nucleoside analogues with the (2-hydroxy-1-phenylethoxy)methyl glycone - A family of nucleoside analogues related to d4T and aciclovir
화학 물질
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(S)-[2-(methoxymethoxy)-2-phenyl]ethyl benzoate
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Identification of a new biaryl scaffold generating potent renin inhibitors
화학 물질
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1,3-dichloro-2-{2-[4-(iodomethyl)phenoxy]ethoxy}-5-methylbenzene
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Synthesis and in vitro and in vivo structure-activity relationships of novel antifungal triazoles for dermatology
화학 물질
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2-(2,4-Difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)-1,2-propanediol
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Development of tryptase inhibitors derived from thalidomide
화학 물질
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2-(4-fluorophenyl)-5-hydroxyisoindole-1,3-dione
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Design and modular parallel synthesis of a MCR derived α-helix mimetic protein-protein interaction inhibitor scaffold
화학 물질
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5-[이소시아노-(톨루엔-4-술포닐)-메틸]-벤조[1,3]디옥솔
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PK/PD Disconnect Observed with a Reversible Endothelial Lipase Inhibitor
화학 물질
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(SS,E)-N-(3-(3,4-dichlorophenyl)propylidene)-2-methylpropane-2-sulfinamide
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A double prodrug system for colon targeting of benzenesulfonamide COX-2 inhibitors
화학 물질
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2-hydroxy-5-(2-{3-oxo-3-[4-(5-p-tolyl-3-trifluoromethyl-pyrazol-1-yl)-benzenesulfonylamino]-propyl}-phenylazo)benzoic acid
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